Table of Contents:
  • What is Pharmacology?
  • How Different Tissues Process Drug Response
  • Drug Receptor Theory
  • Pharmacological Assay Formats: Binding
  • Agonists: The Measurement of Affinity and Efficacy in Functional Assays
  • Orthosteric Drug Antagonism
  • Allosteric Drug Antagonism
  • The Process of Drug Discovery
  • Target- and System-based Strategies for Drug Discovery
  • Hit to Drug: Lead Optimization
  • Statistics and Experimental Design
  • Selected Pharmacological Methods
  • Glossary of Pharmacological Terms
  • Appendices:
  • Statistical Tables
  • Mathematical Fitting Functions.